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化学に関する試験・検査又は研究

Design, synthesis, and biological evaluation of quinazoline derivatives as α-glucosidase inhibitors
Venkateshwarlu Gurram, Ramesh Garlapati, Chiranjeevi Thulluri, Nagaraju Madala, Kumara Swamy Kasani, Pavan Kumar Machiraju, Raju Doddapalla, Uma Addepally, Rambabu Gundla, Balaram Patro, Narender Pottabathini
Medicinal Chemistry Research, DOI: 10.1007/s00044-014-1293-5

First total synthesis of (-)-Auranomide C and its derivatives
Kumaraswamy Sorra, K. Mukkanti and Srinivas Pusuluri
Synthesis 2014, 46, 189-194

Synthesis, anticonvulsant, sedative and anxiolytic activities of novel annulated pyrrolo[1,4]benzodiazepines
Kumaraswamy Sorra, Chi-Fen Chang, Srinivas Pusuluri, Khagga Mukkanti, Min-Chiau Laiu, Bo-Ying Bao, Chia-Hao Su and Ta-Hsien Chuang
International Journal of Molecular Sciences 2014, 15, 16500-16510

A Convenient and Efficient Synthesis of 2-(Het)arylthieno[3,2-b]pyridine-7(4H)-ones and 2,3-Di(het)arylthieno[3,2-b]pyridine-7(4H)-ones
Srinu Puvvala, Vinod D. Jadhav, Sheikh M. Farooq, C. Venkata Ramana Reddy and Pavan Kumar Machiraju
Synthesis 2014; 46(24): 3319-3330

Pyrrolidine and piperidine based chiral spiro and fused scaffolds via build/couple/pair approach
Rajinikanth Mamidala, V. Surendra Babu Damerla, Rambabu Gundla, M. Thirumala Chary, Y. L. N. Murthyd and Subhabrata Sen
RSC Adv., 2014, 4, 10619

Novel Imidazoline Antimicrobial Scaffold That Inhibits DNA Replication with Activity against Mycobacteria and Drug Resistant Gram-Positive Cocci
Kendra K. Harris, Allison Fay, Han-Guang Yan, Pratima Kunwar, Nicholas D. Socci , Narender Pottabathini, Ramakrishna R. Juventhala, Hakim Djaballah, and Michael S. Glickman
ACS Chem. Biol., Article ASAP, DOI: 10.1021/cb500573z, Publication Date: September 15, 2014

Facile total synthesis of gymnoconjugatin A and B
Ramakrishna Samala, Balaram Patro, Manas K. Basu, N. S. Kameswara Rao and K. Mukkanti
Tetrahedron Letters, 2013, 54 (28), 3624–3626

A reagent based DOS strategy via Evans chiral auxiliary: highly stereoselective Michael reaction towards optically active quinolizidinones, piperidinones and pyrrolidinones
Subhabrata Sen, Siva R. Kamma, RambabuGundla, Uma Adepally, Santosh Kuncha, Sridhar Thirnathia and U. Viplava Prasad
RSC. Adv. 2013, 3, 2404

Diversity Oriented Synthesis of Macrocyclic Diaryl Ethers by Dötz Benzannulation
Subhabrata Sen, Rajanikanth Mamidala, Rambabu Gundla and M. T. Charya
Asian J. Org. Chem. 2013, 2, 862 – 868

Synthesis of Privileged Scaffolds by Using Diversity-Oriented Synthesis
Ramu Surakanti, Sumalatha Sanivarapu, Chiranjeevi Thulluri, Pravin S. Iyer, Raghuram S. Tangirala, Rambabu Gundla, Uma Addepally, Y. L. N. Murthy, Lakshmi Velide and Subhabrata Sen
Chem. Asian J. 2013, 8, 1168 – 1176

A novel one-pot synthesis of 7-methoxy-2-arylthieno-[3,2-b]pyridine-3-ols in domino fashion
Srinu Puvvala, Vinod D. Jadhav, Sheikh M. Farooq, Balaram Patro, Ch. Venkata Ramana Reddy
Tetrahedron Letters 54 (2013) 5043–5047

Concise Total Synthesis of (-)-Erinapyrone B from D-(+)-Malic Acid
Ramakrishna Samala, Venkateshwarlu Gurram, Balaram Patroa, Narender Pottabathini & K. Mukkanti
Synthetic Communications, 2013; 44:4, 500-506, DOI: 10.1080/00397911.2013.817017

Development of a-glucosidase inhibitors by room temperature C–C cross couplings of quinazolinones
Ramesh Garlapati, Narender Pottabathini,* Venkateshwarlu Gurram, Kumara Swamy Kasani, Rambabu Gundla, Chiranjeevi Thulluri, Pavan Kumar Machiraju, Avinash B. Chaudhary, Uma Addepally,Raveendra Dayam, Venkata Rao Chunduri and Balaram Patro
Org. Biomol. Chem., 2013, 11, 4778-4791

Ethyl-1-imidazole carbamate (EImC) as a carbonylating agent: Efficient synthesis of oxazolidin-2-ones from amino alcohols.,
R.Venkat Ragavan; Veeraswamy, Somarouthu; Indrasena Reddy, K.; Yennam, Satyanarayana; Jayashree, A..,
Chemistry Letters., 42, 2013, No-2, P109-111

Microwave assisted Westphal condensation and its application to synthesis of sempervirine and related compounds
T. S. Chinta Rao, Sanjay Saha, Gajendra B. Raolji, Balaram Patro, Prabhaker Risbood, Michael J. Difilippantonio, Joseph E. Tomaszewski, Sanjay V. Malhotra,
Tetrahedron Letters 54 (2013) 487–490.

Synthesis and SAR studies of marine natural products ma’edamines A, B and their analogues
Sanjay Saha, Ch. Venkata Ramana Reddy, Shili Xu, Saranya Sankar, Nouri Neamati, Balaram Patro,
Bioorganic & Medicinal Chemistry Letters 23 (2013) 5135–5139.

The first total synthesis and biological evaluation of marine natural products ma’edamines A and B
Sanjay Saha, Ch. Venkata Ramana Reddy, T. Chiranjeevi, Uma Addepally, T. S. Chinta Rao, Balaram Patro,
Bioorganic & Medicinal Chemistry Letters 23 (2013) 1013–1016.

An efficient one-step chemoselective reduction of alkyl ketones over aryl ketones in ß-diketones using LiHMDS and lithium aluminium hydride.
S. Veera Swamy, K. Indrasena Reddy, R. Venkat Ragavan, K. Tirumal Reddy, Satyanarayana Yennam, A. Jayashree.
Tetrahedron Letters., 53, 2012, 4651-4653.

An efficient method for the preparation of mono a-aryl derivatives of diethyl cyanoacetate using ethyl-1-imidazole carbamate (ElmC).
Manoranjan Behera, R.Venkatragavan, M.Sambaiah, Balaiah Erugu, J.Rama Krishna Reddy, K.Mukkanti, Satyanarayana Yennam.
Tetrahedron Letters., 53, (2012), 1060-1062.

Pd-catalyzed amination of 6-halo-2-cyclopropyl-3-(pyridyl-3-ylmethyl) quinazolin-4(3H)-one
Ramesh Garlapati, Narender Pottabathini, Venkateshwarlu Gurram, Avinash B. Chaudhary, Venkata Rao Chunduri, Balaram Patro
Tetrahedron Letters 2012, 53, 5162–5166

Synthesis of novel isoxazole-benzoquinone hybrids via 1,3-dipolar cycloaddition reaction as key step
P. Ravi Kumar, Manoranjan Behera, K. Raghavulu, A. Jaya Shree, Satyanarayana
Tetrahedron Letters 2012, 53, 4108–4113

Synthesis and Cytotoxicity Testing of New Amido-Substituted Triazolopyrrolo[2,1-c][1,4]benzodiazepine (PBDT) Derivatives
Kumaraswamy Sorra, Chi-Fen Chang, Srinivas Pusuluri, Khagga Mukkanti, Min-Chiau Laiu, Bo-Ying Bao, Chia-Hao Su and Ta-Hsien Chuang
Molecules 2012, 17, 8762-8772

C–C Cross-Coupling Reactions of O6-Alkyl-2-Haloinosine Derivatives and a One-Pot Cross-Coupling/O6-Deprotection Procedure
Venkateshwarlu Gurram, Narender Pottabathini*, Ramesh Garlapati, Avinash B. Chaudhary, Balaram Patro, and Mahesh K. Lakshman*
Chemistry-An Asian Journal, 2012, 7(8), 1853-1861

Enantiospecific first total synthesis of 7a(S)-p-hydroxyphenopyrrozin
Yugandhar Kothapalli, Ravi Kumar Puthukanoori, Srinivasa Rao Alapati
Tetrahedron Letters 2012; 53, 1891–1893

Palladium catalyzed synthesis of quinazolino [1,4] benzodiazepine alkaloids and analogues
Kumaraswamy Sorra, Srinivas Pusuluri and K. Mukkanti
Tetrahedron 2012; 68, 2001-2006

Synthesis and Antibacterial Activity of 6-Substituted Anacardic Acid Derivatives
Subhakara Reddy Nallamilli , Ravi Kumar V, Himabindu V, B.Ram and Srinivas Rao Aalapati
Letters in Drug Design & Discovery, 2011, 8, 972-979

Facile two-step synthesis of Crispine A and Harmicine by cyclopropylimine rearrangement
Sanjay Saha, Ch. Venkata Ramana Reddy, Balaram Patro
Tetrahedron Letters, 2011,52, 4014-16

Diversity-oriented synthesis of amino acids using chiral enolates
Subhabrata Sen, Siva R. Kamma, Venkata R. Potti, Y.L.N. Murthy, Avinash B. Chaudhary
Tetrahedron Letters, 2011,52, 5585-5588

Enantioselective synthesis of spirooxoindoles via chiral auxiliary (bicyclic lactam) controlled SNAr reactions
Subhabrata Sen, Venkata R. Potti, Ramu Surakanti, Y. L. N. Murthy and Raghavaiah Pallepogu
Organic & Biomolecular Chemistry, 2011, 9, 626-632

Synthesis and Antibacterial Activity of Anacardic acid derivatives
Subhakara Reddy Nallamilli, Ravi Kumar V, Himabindu.V .B. Ram ,Srinivas Rao Alapati
Letters in Drug Design & Discovery, 2011, 8(7),626-632

SPF32629A and SPF32629B: Enantioselective synthesis, determination of absolute configuration, cytotoxicity and antibacterial evaluation
Srinivasa Rao Vegi, Shanthaveerappa K. Boovanahalli, Balaram Patro, K. Mukkanti
European Journal of Medicinal Chemistry, 2011, 46, 1803-1812

An efficient method for the preparation of mono a-aryl derivatives of diethyl malonate and ethyl cyanoacetate using ethyl-1-imidazole carbamate(EImC)
Manoranjan Behera, R. VenkatRagavan, M. Sambaiah, BalaiahErugu, J. Rama Krishna Reddy, K. Mukkanti, Satyanarayana Yennam
Tetrahedron Letters (December 2011) doi:10.1016/j.tetlet.2011.12.067

Azaindolines: derisking the indoline structural alert
Eugene L. Piatnitski Chekler, Taukeer A. Khan, Rajanikanth Mamidala, James T. Anderson, Raghuram S. Tangirala, Patrick R. Verhoest, Adam M. Gilbert
Article in press, doi:10.1016/j.tetlet.2011.11.070

The first total synthesis of potent human chymase inhibitor SPF32629B via
regioselective bromination and O-acylation strategy
Srinivasa Rao Vegi, Shanthaveerappa K. Boovanahalli, Balaram Patro, K. Mukkanti
Tetrahedron Letters, 2010,51, 2768-2770

Structure-Based Design of 3-Aryl-6-amino-triazolo[4,3-b] pyridazine Inhibitors of Pim-1 Kinase
Ron Grey, Guy W. Bemis, Marc D. Jacobs, Cameron Stuver-Moody, Rahul Jajoo, Narinder Mohal, Jeremy Green
BMCL(Bioorganic & Medicinal Chemistry Letters), 2009, 19(11), 3019-3022

Analytical study of charge transfer complexation of rabeprazole with 2,3-dichloro-5,6-dicyano-1,4-benzoquinone
Nadeem A. Khan, Avinash B. Chaudhary,Balaram Patro ,A. Devika Rani
Science Asia, 2009, 35(4), 365-371

The first total synthesis of novel human chymase inhibitor
Srinivas Rao Vegi, Shanthaveerappa K. Boovanahalli, Arun Prakash Sharma, K. Mukkanti
Tetrahedron, 2008, 49(44),6297-6299

The influence of drug-like concepts on decision-making in medicinal chemistry
Paul D. Leeson, Brian Springthorpe
Nature reviews: drug discovery, 2007